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Program Wageningen 2018

Download the program here!

Program Thursday April 5th 2018

09:00 Welcome & Coffee
09:40 Opening by Jeroen Cornelissen
09:45
Sir Fraser Stoddart (Northwestern University, USA, Sponsored by Wiley / ChemPubSoc)
Materials Beyond Cyclodextrins : Emergence Opens up a Whole New World of Wonders
     
Parallelsession I
(Ir. Haakzaal)
Chair: Romano Orru
Parallelsession II
(Tarthorstzaal)
Chair: Tom Wennekes
10:45
Jordy M. Saya (VU)
HFIP as a Novel Acid Component in the Passerini Reaction: One-Pot Access to β-Amino Alcohols
Marta Artola (UL)
Rational Design of Mechanism-based Retaining Glycosidase Inhibitors
11:05
Luuk Steemers (UvA)
Terephthalic acid derivatives as covalent templates for the synthesis of mechanically interlocked molecules
Johan Pijnenborg (RU)
New chemical tools to modulate sialic acid expression and signaling
11:25
Nabil Tahiri (RUG)
Total synthesis of Mycolic Acids from Mycobacterium tuberculosis for structure elucidation
Dennis Wander (UL)
Doxorubicin and Aclarubicin: Shuffling Glycans for Improved Cytotoxic Agents
     
11:45 Lunch in Terraszaal (ALV @ 12:15 in Tarthorstzaal)
13:15
Keith Woerpel (New York University, USA, Sponsored by Mettler-Toledo)
Stereoselective Addition Reactions to Carbon Electrophiles: Conformational Analysis, Stereoelectronic Effects, and Reactivity
     
Parallelsession III
(Ir. Haakzaal)
Chair: Mark Borst
Parallelsession IV
(Tarthorstzaal)
Chair: Kim Bonger
14:15
Hidde Elferink (RU)
Glycosylations Caught in the Act
Can Araman (UL)
Amyloid-like behavior of citrullinated myelin oligodendrocyte protein (MOG) derived epitope peptides lead to enhanced antigen presentation in multiple sclerosis
14:35
J. Braun (VU)
Intramolecular Tsuji-Trost Cascade Cyclization to Fused Vinylcyclopropanes
Niek van der Zouwen (RUG)
In Situ Combinatorial Synthesis and Screening of Chemical Probes
14:55
Stella Verkhnyatskaya (RUG)
Fucosylated Cyclodextrins as Novel Antiadhesives
Jorick Bruins (WUR)
Inducible, selective labelling of antibodies via enzymatic oxidation of tyrosine to 1,2-quinones
   
15:15 Coffee/Tea in Terraszaal
15:45
Annemiek Madder (Ghent University, BE, Sponsored by Elsevier)
Furan-based Click and Photo-click Reactions for the Study and Targeting of Protein and Nucleic Acid Interactions
16:45
Laura Kiessling (Massachusetts Institute of Technology, USA, Sponsored by Screening Devices)
Glycans as Cellular IDs
17:45
Announcement of 2017 winner 'The KNCV - Dr. J.H. Backer Organic Chemsitry Award'
18:00 Dinner (registration necessary)

 

Program Friday April 6th 2018

09:15 Coffee in Terraszaal
09:45
David Spring (University of Cambridge, UK, Sponsored by ChemConnection part of Ardena)
Enriching Chemical Space to Drug Undruggable Targets
     
Parallelsession V
(Ir. Haakzaal)
Chair: Gino van Strijdonck
Parallelsession VI
(Tarthorstzaal)
Chair: Leendert van den Bos
10:45
Pia Kröger (UT)
Versatile Single Chain Polymeric Nanoparticles via Thiol-Michael Addition
Reinder de Vries (RUG)
Bio-orthogonal Chemical Modification of Peptide Antibiotics
11:05
Jaime Mateos (RUG)
Regio- and Stereoselective Synthesis of Borylated 1,4-Dienes by Cu/Pd Dual Catalysis
Mark A.R. de Geus (UL)
Chemical Control over T-Cell Activation In Vivo Using Deprotection of Trans-cyclooctene-modified Epitopes
11:25
Sybrin Schröder (UL)
Activity-based protein profiling of exo- and endo-xylanases in Aspergillus secretomes
Seino Jonkees (UU)
Macrocyclic peptide inhibitors of carbohydrate-active enzymes
   
11:45 Lunch in Terraszaal
13:00
Roeland Nolte (Radboud University, NL)
Encoding polymers with information. A supramolecular approach
     
Parallelsession VII
(Ir. Haakzaal)
Chair: Romano Orru
Parallelsession VIII
(Tarthorstzaal)
Chair: Tom Wennekes
13:45
Flip Holtrop (UvA)
Van der Waals forces in frustrated Lewis pair chemistry
Digvijay Gahtory (WUR)
New click on the block: Strain‐promoted cycloaddition of cyclopropenes with o‐quinones
14:05
Shuqin Cao (UT)
Supramolecular Chemistry Inside Protein Cages
Victor J. Somovilla (UU)
Fluoroproline in MUC1 antigen opens a new via in the development of enhanced cancer diagnostic tools
   
14:25 Coffee/Tea in Terraszaal
15:00
Rachel O’Reilly (University of Birmingham, UK, Sponsored by Buchi)
Semi-crystalline polymers for controlled self-assembly
16:00
MG Finn (Georgia Institute of Technology, USA, Sponsored by MercachemSyncom)
Click, Carry, and Release: Building and Transporting Molecular Function
17:00 Closing followed by drinks @ Down under bar
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